SCHEMBL6201040

SCHEMBL6201040

O=C(NC(=O)C1CCNCC1)c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
P2RY14 Q15391 1/20 0.46
KDM4E B2RXH2 3/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 1/20 0.46
MPO P05164 1/20 0.43
CYP1A2 P05177 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CYP2A6 P11509 1/20 0.43
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
ACVRL1 P37023 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
MAPT P10636 1/20 0.40
GSK3B P49841 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203700 0.82 KDM4E (0.45) ALDH1A1KDM4ECYP3A4CYP2D6CYP2C19
SCHEMBL16333620 0.81 KMT2A (0.52) CYP2D6L3MBTL1GSK3B
SCHEMBL4672867 0.78 MEN1 (0.62) ALDH1A1P2RY14KDM4ECYP3A4CYP2D6
SCHEMBL29050693 0.78 L3MBTL1 (0.54) ALDH1A1KDM4EGAAL3MBTL1
SCHEMBL1553389 0.78 ROCK2 (0.61) CYP3A4CYP2D6ACVRL1
Hydrochloric Acid SCHEMBL27414471 0.76 ROCK2 (0.60) CYP3A4CYP2D6ACVRL1
SCHEMBL4629627 0.75 MC4R (0.50) ALDH1A1P2RY14CYP1A2
SCHEMBL4393712 0.74 ALDH1A1 (0.64) ALDH1A1L3MBTL1MAPT
SCHEMBL2004792 0.73 ALDH1A1 (0.73) ALDH1A1KDM4ECYP3A4CYP2D6CYP2C19
SCHEMBL241357 0.72 HDAC4 (0.53) ALDH1A1KDM4EGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed