SCHEMBL6204518

SCHEMBL6204518

NC(=O)[C@@H](C(=O)N(C(=O)c1ccco1)C1CCCNCC1O)C1CCCC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
HPGD P15428 2/20 0.35
POLB P06746 2/20 0.34
CHRNB2 P17787 3/20 0.32
CHRNA7 P36544 3/20 0.32
CHRNA4 P43681 3/20 0.32
CHRNB4 P30926 2/20 0.32
CHRNA3 P32297 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
PKM P14618 1/20 0.31
TP53 P04637 1/20 0.31
CCR5 P51681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203389 0.82 ALDH1A1 (0.34) ALDH1A1HPGDPOLBTSHRTDP1
SCHEMBL6204515 0.75 TSHR (0.31) TSHR
SCHEMBL7493491 0.63 OPRM1 (0.43) ALDH1A1KMT2ACCR5
SCHEMBL6206698 0.63 KDM4E (0.38) MAPTTSHRKMT2ASMN1; SMN2
SCHEMBL5099682 0.63 KMT2A (0.39) KMT2A
SCHEMBL4765023 0.61 CTSD (0.38)
SCHEMBL3285958 0.58 ALDH1A1 (0.53) ALDH1A1HPGDMEN1MAPTTSHR
Piperazine SCHEMBL635835 0.58 CES2 (0.52) ALDH1A1POLBCHRNB2CHRNA7CHRNA4
SCHEMBL12531247 0.58 ALDH1A1 (0.64) ALDH1A1HPGDMEN1TSHRKMT2A
SCHEMBL16475935 0.58 CPN1 (0.47) MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539178-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2005-06-15 EP disclosed
WO-2004017911-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-03-04 WO disclosed