SCHEMBL6204811

SCHEMBL6204811

CCCN(CO)c1nc(NCc2ccc(OC)c(O)c2O)c2[nH]nnc2n1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRUNE1 Q86TP1 1/20 0.32
TSHR P16473 2/20 0.32
HSD17B10 Q99714 2/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 4/20 0.32
MAPT P10636 3/20 0.32
GAA P10253 2/20 0.32
NPC1 O15118 1/20 0.32
ALOX12 P18054 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PKM P14618 1/20 0.31
HTT P42858 2/20 0.31
KDM4E B2RXH2 1/20 0.31
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
PDE5A O76074 1/20 0.31
PDE6C P51160 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204808 0.86 PRUNE1 (0.37) PRUNE1TSHRHSD17B10SMN1; SMN2ALDH1A1
SCHEMBL6205414 0.85 HMGCR (0.32) PRUNE1
SCHEMBL6203855 0.83 CCNE1 (0.34) PRUNE1TSHRHSD17B10TP53SMN1; SMN2
SCHEMBL6203495 0.80 PRUNE1 (0.35) PRUNE1CCNE1CDK2PDE5APDE6C
SCHEMBL6203171 0.79 CCNE1 (0.37) CCNE1CDK2
SCHEMBL6202760 0.79 CDK1 (0.40) PRUNE1TSHRSMN1; SMN2CCNE1CDK2
SCHEMBL6204719 0.78 PGK1 (0.33)
SCHEMBL3444717 0.76 CDK2 (0.52) TSHRTP53SMN1; SMN2ALDH1A1RAB9A
SCHEMBL3445281 0.75 CDK2 (0.38) HSD17B10ALDH1A1MAPTGAANPC1
SCHEMBL3445936 0.74 CDK1 (0.41) MAPTRAB9APKMKDM4ECCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed