SCHEMBL6207527

SCHEMBL6207527

CC(=O)N1CCN(S(=O)(=O)c2ccccc2)C(C(=O)NS(=O)(=O)Cc2ccc3c(c2)OCO3)C1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
MAPT P10636 2/20 0.49
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MMP1 P03956 3/20 0.45
MMP9 P14780 3/20 0.45
MMP13 P45452 3/20 0.45
MMP3 P08254 2/20 0.45
MMP7 P09237 2/20 0.45
ADAM17 P78536 1/20 0.44
HTT P42858 1/20 0.43
GAA P10253 2/20 0.43
USP2 O75604 1/20 0.43
PKM P14618 1/20 0.43
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033190 0.88 MAPT (0.65) ALDH1A1MAPTMEN1KMT2AHTT
SCHEMBL4032764 0.74 MMP1 (0.62) ALDH1A1MMP1MMP9MMP13MMP3
SCHEMBL2440987 0.70 FKBP1A (0.53) ALDH1A1MMP1MMP9MMP13MMP3
SCHEMBL7346677 0.70 MMP1 (0.54) ALDH1A1MEN1KMT2AMMP1MMP9
SCHEMBL4032527 0.69 USP2 (0.60) ALDH1A1MMP1MMP9MMP13MMP3
SCHEMBL4033188 0.68 ALDH1A1 (0.46) ALDH1A1MAPTMEN1KMT2AHTT
SCHEMBL26848353 0.67 L3MBTL1 (0.62) ALDH1A1MEN1KMT2AMMP1MMP9
SCHEMBL2437981 0.67 MMP1 (0.58) ALDH1A1MMP1MMP9MMP13MMP3
SCHEMBL6237734 0.67 MMP1 (0.71) MMP1MMP9MMP13MMP3MMP7
SCHEMBL4402232 0.66 MMP1 (0.78) MMP1MMP9MMP13MMP3MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2005-11-09 EP disclosed
WO-2004071390-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-08-26 WO disclosed