SCHEMBL6208321

SCHEMBL6208321

CCOC(=O)C#CC1(O)CCN(C(=O)OCC(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
TSHR P16473 2/20 0.37
ALDH1A1 P00352 5/20 0.36
POLB P06746 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 1/20 0.36
HRH2 P25021 2/20 0.35
HRH1 P35367 2/20 0.35
GAA P10253 3/20 0.35
RECQL P46063 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
RAB9A P51151 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
KIT P10721 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693197 0.81 USP2 (0.40) L3MBTL1TSHRSMN1; SMN2
SCHEMBL3956031 0.79 JAK2 (0.37) L3MBTL1TSHRHRH2HRH1CYP2D6
SCHEMBL3955003 0.78 CYP2D6 (0.39) L3MBTL1TSHRHRH2HRH1GAA
SCHEMBL8867607 0.77 L3MBTL1 (0.45) L3MBTL1TSHRALDH1A1POLBSMN1; SMN2
SCHEMBL7096473 0.74 TLR8 (0.35) L3MBTL1ALDH1A1SMN1; SMN2GAA
SCHEMBL8866898 0.73 L3MBTL1 (0.41) L3MBTL1TSHRALDH1A1POLBSMN1; SMN2
SCHEMBL6824028 0.71 ALDH1A1 (0.50) L3MBTL1TSHRALDH1A1POLBSMN1; SMN2
SCHEMBL3663186 0.70 CYP2D6 (0.42) L3MBTL1TSHRALDH1A1HRH2HRH1
SCHEMBL4074787 0.70 RAB9A (0.41) L3MBTL1ALDH1A1HRH2HRH1CYP2D6
SCHEMBL26705603 0.69 RAB9A (0.40) L3MBTL1TSHRALDH1A1CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603901-A1 TETRAHYDROPYRAN COMPOUNDS AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 2005-12-14 EP disclosed
WO-2004078750-A1 TETRAHYDROPYRAN COMPOUNDS AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 2004-09-16 WO disclosed