SCHEMBL6208514

SCHEMBL6208514

CC(C)C[C@@H](C(N)=O)N(CC#N)c1nscc1Br

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208765 0.79 CTSL (0.36) CTSLCTSBCTSS
SCHEMBL4701834 0.77 CTSB (0.39) CTSLCTSBCTSS
SCHEMBL6208510 0.77 CTSB (0.39) CTSLCTSBCTSS
SCHEMBL4703744 0.75 KDM4E (0.36) CTSLCTSBCTSS
SCHEMBL4703503 0.75 KDM4E (0.36) CTSLCTSBCTSS
SCHEMBL4703890 0.72 CTSS (0.40) CTSLCTSBCTSS
SCHEMBL4704327 0.72 CTSL (0.51) CTSLCTSBCTSS
SCHEMBL4698962 0.72 CTSL (0.37) CTSLCTSBCTSS
SCHEMBL4704891 0.71 CTSL (0.37) CTSLCTSBCTSS
SCHEMBL4701851 0.71 CTSL (0.49) CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-A4 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-10-12 EP disclosed
EP-1372655-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada & Co. (CA) 2004-01-02 EP disclosed
WO-2002069901-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2002-09-12 WO disclosed