SCHEMBL6209614

SCHEMBL6209614

CC(CCNC(=O)c1ccc(-n2ccnc2)cc1)CC(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.41
CYP4Z1 Q86W10 1/20 0.38
ADRB1 P08588 4/20 0.37
DRD3 P35462 5/20 0.37
DRD2 P14416 4/20 0.37
AHR P35869 1/20 0.36
ADRB2 P07550 3/20 0.35
ADRB3 P13945 3/20 0.35
TAOK1 Q7L7X3 1/20 0.35
TAOK3 Q9H2K8 1/20 0.35
GFER P55789 1/20 0.35
DNMT3B Q9UBC3 1/20 0.35
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210874 0.89 ALDH1A1 (0.40) NAMPT
SCHEMBL6211167 0.89 CTSK (0.39) DRD3
SCHEMBL6209043 0.89 LMNA (0.41)
SCHEMBL6210327 0.87 GAA (0.45)
SCHEMBL6212088 0.87 SLC6A5 (0.40) NAMPT
SCHEMBL6259636 0.87 HDAC3 (0.35) NAMPT
SCHEMBL6209727 0.86 CHRM4 (0.42)
SCHEMBL6210258 0.85 POLB (0.42)
SCHEMBL6211027 0.85 NAMPT (0.40) NAMPT
SCHEMBL6210236 0.84 CHRM4 (0.41) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed