SCHEMBL4046533

SCHEMBL4046533

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)Oc1cccc2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CTSK P43235 3/20 0.35
ACE P12821 2/20 0.35
ACE2 Q9BYF1 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
GPR132 Q9UNW8 3/20 0.33
MC4R P32245 1/20 0.33
MC3R P41968 1/20 0.33
MC1R Q01726 1/20 0.33
F12 P00748 1/20 0.33
CYP51A1 Q16850 1/20 0.33
CMKLR2 P46091 1/20 0.33
CMKLR1 Q99788 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6212077 0.90 CTSL (0.39) POLBCTSKACEACE2CTSB
SCHEMBL4049549 0.88 GPR132 (0.38) CTSKACEACE2CTSBCTSS
SCHEMBL4042676 0.87 CTSB (0.36) MAPK1ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL4041433 0.86 ALDH1A1 (0.35) ALDH1A1POLBCTSBCTSSMC4R
SCHEMBL4047478 0.84 MC4R (0.37) CTSKACECTSBCTSSMC4R
SCHEMBL4043722 0.84 CTSK (0.40) CTSKACEACE2CTSBCTSS
SCHEMBL6209627 0.83 CHRNB2 (0.42) MAPTCTSKACEACE2CTSB
SCHEMBL4040214 0.83 GPR132 (0.39) SMN1; SMN2CTSKACEGPR132MC4R
SCHEMBL4042165 0.82 EPHX1 (0.37) CTSKACECTSBCTSSGPR132
SCHEMBL4041149 0.81 ITGA4 (0.39) ALDH1A1MAPTCTSKACEITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed