SCHEMBL4049549

SCHEMBL4049549

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 4/20 0.38
CTSK P43235 3/20 0.38
ECE1 P42892 1/20 0.37
ACE P12821 2/20 0.37
CHRNA7 P36544 1/20 0.37
ACE2 Q9BYF1 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CMKLR2 P46091 1/20 0.35
CMKLR1 Q99788 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
MMP12 P39900 1/20 0.35
ITGA4 P13612 2/20 0.35
ITGB7 P26010 2/20 0.35
ADAM17 P78536 1/20 0.35
EPHX1 P07099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041149 0.94 ITGA4 (0.39) CTSKECE1ACECHRNA7MMP12
SCHEMBL4040214 0.94 GPR132 (0.39) GPR132CTSKECE1ACECHRNA7
SCHEMBL4042165 0.93 EPHX1 (0.37) GPR132CTSKECE1ACECHRNA7
SCHEMBL4045083 0.89 CTSK (0.47) CTSKCHRNA7CTSBCTSSEPHX1
SCHEMBL4047771 0.89 CTSK (0.39) GPR132CTSKECE1CHRNA7ADAM17
SCHEMBL4046533 0.88 MAPK1 (0.36) GPR132CTSKACEACE2CTSB
SCHEMBL4047615 0.87 CTSB (0.38) GPR132CTSKECE1ACECHRNA7
SCHEMBL4046868 0.85 ITGB1 (0.37) GPR132CTSKACE2CTSBCTSS
SCHEMBL4042529 0.84 BCL2 (0.38) GPR132CTSKACECMKLR2CMKLR1
SCHEMBL4043883 0.83 CTSK (0.42) CTSKACEACE2CTSSITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed