SCHEMBL6210489

SCHEMBL6210489

CC(CCNC(=O)c1ccc(-c2cccs2)cc1)CC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.39
DRD4 P21917 6/20 0.37
DRD2 P14416 5/20 0.37
HTR2A P28223 4/20 0.37
DPP4 P27487 1/20 0.37
PREP P48147 1/20 0.37
HDAC1 Q13547 4/20 0.36
FYN P06241 1/20 0.36
SMYD3 Q9H7B4 2/20 0.35
LMNA P02545 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211053 0.90 CHRM4 (0.39) CHRM4DRD4DRD2HTR2ADPP4
SCHEMBL6211570 0.89 SLC6A5 (0.38) CHRM4SMYD3LMNA
SCHEMBL6210236 0.88 CHRM4 (0.41) CHRM4DRD4DRD2HTR2ADPP4
SCHEMBL6210587 0.88 HDAC1 (0.42) CHRM4DRD4DRD2HTR2ADPP4
SCHEMBL6208718 0.88 LMNA (0.42) CHRM4SMYD3LMNA
SCHEMBL6209295 0.88 CTSK (0.37) HTR2AHDAC1SMYD3LMNAHDAC3
SCHEMBL6211038 0.88 CTSK (0.41) SMYD3LMNA
SCHEMBL6209450 0.88 CXCR3 (0.43) CHRM4SMYD3LMNA
SCHEMBL6209104 0.87 CHRM4 (0.41) CHRM4DRD4DRD2HTR2ADPP4
SCHEMBL6210230 0.87 ROCK2 (0.40) SMYD3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed