SCHEMBL6235518

SCHEMBL6235518

O=C(c1ccnc(C(=O)N(CCc2ccc(Cl)cc2)CCc2ccc(Cl)cc2)c1)N(CCc1ccc(Cl)cc1)CCc1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
SLC2A1 P11166 1/20 0.40
C5AR1 P21730 1/20 0.40
PTGIR P43119 2/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA9 Q16790 1/20 0.38
LPAR1 Q92633 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235516 0.92 KDM4C (0.49) ALDH1A1MAPTL3MBTL1PSEN1PSEN2
SCHEMBL6239726 0.86 ALDH1A1 (0.46) ALDH1A1MAPTL3MBTL1NPC1RAB9A
SCHEMBL6985934 0.86 MAPT (0.43) ALDH1A1MAPTL3MBTL1PSEN1PSEN2
SCHEMBL6991899 0.86 MAPT (0.51) ALDH1A1MAPTL3MBTL1PSEN1PSEN2
SCHEMBL6989792 0.86 MEN1 (0.45) ALDH1A1MAPTL3MBTL1NPC1RAB9A
SCHEMBL6990114 0.83 LPAR1 (0.49) ALDH1A1SLC2A1CA12CA1CA2
SCHEMBL6985928 0.79 KDM5B (0.49) ALDH1A1MAPTL3MBTL1KDM4EKDM6B
SCHEMBL6239722 0.79 KDM5B (0.49) ALDH1A1MAPTL3MBTL1LPAR1LPAR5
SCHEMBL6993032 0.79 KMT2A (0.49) ALDH1A1CA12CA1CA2CA9
SCHEMBL6985002 0.78 KDM4E (0.42) ALDH1A1MAPTL3MBTL1LPAR1LPAR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed