SCHEMBL6239726

SCHEMBL6239726

CCc1ccc(CCN(CCc2ccc(CC)cc2)C(=O)c2ccnc(C(=O)N(CCc3ccc(CC)cc3)CCc3ccc(CC)cc3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
MAPT P10636 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPK1 P28482 1/20 0.38
KDM4C Q9H3R0 3/20 0.37
KDM5A P29375 2/20 0.37
KDM5B Q9UGL1 2/20 0.37
KDM4E B2RXH2 1/20 0.37
KDM6B O15054 1/20 0.37
TET3 O43151 1/20 0.37
KDM4A O75164 1/20 0.37
BBOX1 O75936 1/20 0.37
KDM5C P41229 1/20 0.37
ASPH Q12797 1/20 0.37
KDM4D Q6B0I6 1/20 0.37
TET2 Q6N021 1/20 0.37
ALKBH5 Q6P6C2 1/20 0.37
KDM7A Q6ZMT4 1/20 0.37
KDM8 Q8N371 1/20 0.37
TET1 Q8NFU7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6239722 0.92 KDM5B (0.49) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6985934 0.89 MAPT (0.43) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6235518 0.86 ALDH1A1 (0.49) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6989792 0.86 MEN1 (0.45) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6990114 0.86 LPAR1 (0.49) ALDH1A1CA12CA1CA2CA9
SCHEMBL16569986 0.83 ALDH1A1 (0.53) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6985928 0.82 KDM5B (0.49) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6993032 0.81 KMT2A (0.49) ALDH1A1MAPK1KDM4ECA12CA1
SCHEMBL5808527 0.79 ALDH1A1 (0.69) ALDH1A1MAPTL3MBTL1KDM4CKDM5A
SCHEMBL6989317 0.79 SMN1; SMN2 (0.47) MAPTCA1CA2CA9NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed