SCHEMBL6993032

SCHEMBL6993032

COc1ccc(CCN(CCc2ccc(OC)c(OC)c2)C(=O)c2ccnc(C(=O)N(CCc3ccc(OC)c(OC)c3)CCc3ccc(OC)c(OC)c3)c2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
CYP3A4 P08684 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
LMNA P02545 2/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
AOC3 Q16853 1/20 0.46
KDM4E B2RXH2 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPK1 P28482 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
ELANE P08246 1/20 0.44
PKM P14618 1/20 0.44
CDK8 P49336 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993029 0.93 ALDH1A1 (0.48) KMT2ACYP3A4ALDH1A1MEN1CYP1A2
SCHEMBL6990114 0.85 LPAR1 (0.49) KMT2ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL6986949 0.82 SLC2A1 (0.48) AOC3
SCHEMBL6239726 0.81 ALDH1A1 (0.46) ALDH1A1KDM4EMAPK1CA12CA1
SCHEMBL6985934 0.81 MAPT (0.43) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL6235518 0.79 ALDH1A1 (0.49) ALDH1A1CYP1A2LMNAKDM4ECA12
SCHEMBL6990109 0.79 LPAR1 (0.53) KMT2ACYP3A4ALDH1A1MEN1KDM4E
SCHEMBL6989792 0.78 MEN1 (0.45) KMT2AALDH1A1MEN1LMNAKDM4E
SCHEMBL6989317 0.77 SMN1; SMN2 (0.47) CYP3A4CYP2D6LMNASMN1; SMN2CA1
SCHEMBL18864231 0.77 MAPT (0.46) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362033-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP claimed
WO-2002064568-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed