SCHEMBL6235626

SCHEMBL6235626

O=C(c1ccnc(C(=O)N(Cc2ccccc2-c2ccccc2)Cc2ccccc2-c2ccccc2)c1)N(Cc1ccccc1-c1ccccc1)Cc1ccccc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 8/20 0.47
KMT2A Q03164 1/20 0.39
KCNA5 P22460 1/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
KDM6B O15054 1/20 0.39
TET3 O43151 1/20 0.39
KDM4A O75164 1/20 0.39
BBOX1 O75936 1/20 0.39
KDM5A P29375 1/20 0.39
KDM5C P41229 1/20 0.39
ASPH Q12797 1/20 0.39
KDM4D Q6B0I6 1/20 0.39
TET2 Q6N021 1/20 0.39
ALKBH5 Q6P6C2 1/20 0.39
KDM7A Q6ZMT4 1/20 0.39
KDM8 Q8N371 1/20 0.39
TET1 Q8NFU7 1/20 0.39
EGLN2 Q96KS0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235628 0.94 KDM4C (0.48) GPBAR1KMT2AALDH1A1MAPTKDM4E
SCHEMBL6989757 0.82 MAPT (0.47) KMT2AALDH1A1MAPTKDM4EKDM4A
SCHEMBL6989518 0.82 ALDH1A1 (0.46) KMT2AALDH1A1MAPTKDM4AKDM5A
SCHEMBL6987326 0.82 ALDH1A1 (0.43) KMT2AALDH1A1MAPTKDM4EKDM6B
SCHEMBL5210605 0.81 CFTR (0.55) KMT2AALDH1A1MAPTKDM4EKDM6B
SCHEMBL6985789 0.80 HDAC1 (0.51) ALDH1A1MAPTKDM4EKDM4AKDM4C
SCHEMBL6988723 0.79 SMN1; SMN2 (0.47) KMT2AALDH1A1MAPTKDM4EKDM4A
SCHEMBL6985787 0.75 KDM4A (0.50) ALDH1A1MAPTKDM4EKDM6BTET3
SCHEMBL5210601 0.74 KDM4E (0.56) KMT2AALDH1A1MAPTKDM4EKDM6B
SCHEMBL5214358 0.74 PPARG (0.55) KMT2AALDH1A1MAPTHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed