SCHEMBL6989518

SCHEMBL6989518

O=C(c1ccnc(C(=O)N(Cc2ccccc2Cl)Cc2ccccc2Cl)c1)N(Cc1ccccc1Cl)Cc1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
MAPT P10636 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
RAF1 P04049 1/20 0.44
MAP2K1 Q02750 1/20 0.44
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
TP53 P04637 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4C Q9H3R0 2/20 0.40
KDM5B Q9UGL1 2/20 0.40
THRB P10828 1/20 0.40
KDM5A P29375 1/20 0.40
KMT2A Q03164 2/20 0.39
ANO1 Q5XXA6 2/20 0.39
HTT P42858 1/20 0.39
KDM4A O75164 1/20 0.38
MEN1 O00255 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987326 0.84 ALDH1A1 (0.43) ALDH1A1MAPTL3MBTL1CYP1A2CYP3A4
SCHEMBL6989757 0.84 MAPT (0.47) ALDH1A1MAPTL3MBTL1TP53SMN1; SMN2
SCHEMBL6985789 0.82 HDAC1 (0.51) ALDH1A1MAPTL3MBTL1CYP1A2CYP2C19
SCHEMBL6235626 0.82 GPBAR1 (0.47) ALDH1A1MAPTL3MBTL1KDM4CKDM5B
SCHEMBL6988723 0.81 SMN1; SMN2 (0.47) ALDH1A1MAPTRAF1MAP2K1CYP1A2
SCHEMBL5210605 0.80 CFTR (0.55) ALDH1A1MAPTL3MBTL1KDM4CKDM5B
SCHEMBL6991899 0.78 MAPT (0.51) ALDH1A1MAPTL3MBTL1TP53KDM4C
SCHEMBL6236957 0.77 MAPT (0.51) ALDH1A1MAPTL3MBTL1SMN1; SMN2KDM4C
SCHEMBL6235628 0.75 KDM4C (0.48) ALDH1A1MAPTKDM4CKDM5BKDM5A
SCHEMBL6985787 0.74 KDM4A (0.50) ALDH1A1MAPTCYP1A2CYP2C19KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362033-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP claimed
WO-2002064568-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed