SCHEMBL6988723

SCHEMBL6988723

COc1ccccc1CN(Cc1ccccc1OC)C(=O)c1ccnc(C(=O)N(Cc2ccccc2OC)Cc2ccccc2OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 2/20 0.45
TP53 P04637 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
POLB P06746 1/20 0.44
ACHE P22303 2/20 0.43
TSHR P16473 3/20 0.43
KDM4A O75164 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
NPC1 O15118 1/20 0.42
BCHE P06276 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TSPO P30536 1/20 0.42
RAF1 P04049 1/20 0.42
MAP2K1 Q02750 1/20 0.42
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987326 0.83 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL6989518 0.81 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1MAPTTP53MEN1
SCHEMBL6989757 0.81 MAPT (0.47) SMN1; SMN2ALDH1A1KDM4EMAPTTP53
SCHEMBL6235626 0.79 GPBAR1 (0.47) ALDH1A1KDM4EMAPTKMT2AKDM4A
SCHEMBL6985789 0.79 HDAC1 (0.51) SMN1; SMN2ALDH1A1KDM4EMAPTKDM4A
SCHEMBL5210605 0.77 CFTR (0.55) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL11900421 0.77 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1KDM4EMAPTTP53
SCHEMBL6990533 0.77 SLC2A1 (0.53) ALDH1A1MAPTMEN1KMT2ATSHR
SCHEMBL6990355 0.77 SLC2A1 (0.61) SMN1; SMN2POLB
SCHEMBL6989554 0.74 HRH1 (0.41) MAPTTSHRKDM4CRAF1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362033-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP claimed
WO-2002064568-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed