SCHEMBL6987326

SCHEMBL6987326

Cc1ccccc1CN(Cc1ccccc1C)C(=O)c1ccnc(C(=O)N(Cc2ccccc2C)Cc2ccccc2C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 7/20 0.41
HSD17B10 Q99714 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
PKM P14618 1/20 0.40
ALKBH2 Q6NS38 1/20 0.40
ALKBH3 Q96Q83 1/20 0.40
OPRK1 P41145 3/20 0.40
KDM4A O75164 2/20 0.40
KDM5A P29375 2/20 0.40
KDM4C Q9H3R0 2/20 0.40
KDM5B Q9UGL1 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6232235 0.87 KDM4A (0.43) ALDH1A1L3MBTL1MAPTKDM4EHSD17B10
SCHEMBL6989757 0.84 MAPT (0.47) ALDH1A1L3MBTL1MAPTKDM4EKMT2A
SCHEMBL6989518 0.84 ALDH1A1 (0.46) ALDH1A1L3MBTL1MAPTKMT2AMEN1
SCHEMBL6988723 0.83 SMN1; SMN2 (0.47) ALDH1A1MAPTKDM4EKMT2AMEN1
SCHEMBL6985789 0.82 HDAC1 (0.51) ALDH1A1L3MBTL1MAPTKDM4EHSD17B10
SCHEMBL6235626 0.82 GPBAR1 (0.47) ALDH1A1L3MBTL1MAPTKDM4EKMT2A
SCHEMBL5210605 0.80 CFTR (0.55) ALDH1A1L3MBTL1MAPTKDM4EKMT2A
SCHEMBL6232231 0.80 KDM4A (0.52) ALDH1A1L3MBTL1MAPTKDM4EALKBH2
SCHEMBL6992829 0.78 MAPT (0.46) ALDH1A1L3MBTL1MAPTKDM4EKMT2A
SCHEMBL5808527 0.76 ALDH1A1 (0.69) ALDH1A1L3MBTL1MAPTKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362033-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP claimed
WO-2002064568-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed