SCHEMBL6236087

SCHEMBL6236087

O=C(NC(CC1CC1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)c1cc2sccc2s1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.35
CTSV O60911 2/20 0.34
CTSL P07711 2/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.34
F2 P00734 4/20 0.33
GPR132 Q9UNW8 1/20 0.33
HTRA1 Q92743 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
GCK P35557 1/20 0.32
FKBP1A P62942 1/20 0.32
F10 P00742 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044323 0.90 SMYD3 (0.33) SMYD3F2GPR132GCKFKBP1A
SCHEMBL4040540 0.83 CTSK (0.51) SMYD3CTSVCTSLCTSSCTSK
SCHEMBL4043646 0.83 CTSS (0.38) SMYD3CTSVCTSLCTSSCTSK
SCHEMBL4045303 0.82 CTSK (0.37) SMYD3CTSLCTSSCTSKALDH1A1
SCHEMBL4045954 0.82 SMYD3 (0.33) SMYD3CTSSCTSKALDH1A1FKBP1A
SCHEMBL4044199 0.82 SMYD3 (0.34) SMYD3F2ALDH1A1FKBP1AF10
SCHEMBL6238658 0.81 HSD17B10 (0.37) SMYD3CTSKALDH1A1GAA
SCHEMBL4042255 0.81 CTSS (0.42) CTSVCTSLCTSSCTSKGPR132
SCHEMBL4045457 0.80 FKBP1A (0.39) SMYD3ALDH1A1FKBP1A
SCHEMBL4051011 0.80 HCRTR2 (0.34) SMYD3CTSVCTSLCTSSGCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed