SCHEMBL6237020

SCHEMBL6237020

COc1ccc(CNc2nc(C#N)nc(Nc3ccccc3)n2)cc1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.58
KCNH3 Q9ULD8 3/20 0.56
ADORA2A P29274 1/20 0.55
ADORA2B P29275 1/20 0.55
SLC2A1 P11166 2/20 0.55
CTSK P43235 2/20 0.54
CTSL P07711 1/20 0.54
CTSS P25774 1/20 0.54
MAPT P10636 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3289406 0.90 KCNH3 (0.69) KCNH3SLC2A1MAPTNPSR1L3MBTL1
SCHEMBL13325954 0.80 APP (0.67) KCNH3SLC2A1MAPTNPSR1L3MBTL1
SCHEMBL13363711 0.79 TDP1 (0.70) TDP1KCNH3ADORA2ACTSK
SCHEMBL6235242 0.78 CTSK (0.76) TDP1ADORA2ACTSKMAPT
SCHEMBL3287006 0.77 CTSL (0.61) KCNH3SLC2A1CTSKCTSLCTSS
SCHEMBL10073747 0.77 KCNH3 (0.77) TDP1KCNH3ADORA2AADORA2BSLC2A1
SCHEMBL10099686 0.77 KCNH3 (0.77) TDP1KCNH3ADORA2AADORA2BSLC2A1
SCHEMBL6237210 0.77 TDP1 (0.75) TDP1KCNH3CTSK
SCHEMBL6237023 0.76 ADORA2A (0.53) ADORA2AADORA2BCTSKCTSLCTSS
SCHEMBL6234331 0.76 CTSK (0.68) TDP1KCNH3CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011703-A1 2-CYANO-1,3,5-TRIAZINE-4,6-DIAMINE DERIVATIVES AKZO NOBEL N.V. (NL) 2005-02-10 WO disclosed