SCHEMBL6237023

SCHEMBL6237023

COc1ccc(N(C)c2nc(C#N)nc(Nc3ccccc3)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.53
ADORA2B P29275 2/20 0.53
CTSK P43235 5/20 0.49
CTSL P07711 4/20 0.49
CTSS P25774 4/20 0.49
CTSB P07858 3/20 0.47
CDK1 P06493 1/20 0.47
KDR P35968 1/20 0.47
MERTK Q12866 1/20 0.47
NPY5R Q15761 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14264146 0.83 ALDH1A1 (0.52) ADORA2AADORA2BKDRMERTKNPY5R
SCHEMBL17220082 0.76 LMNA (0.50) ADORA2AKDRMERTK
SCHEMBL6237020 0.76 TDP1 (0.58) ADORA2AADORA2BCTSKCTSLCTSS
SCHEMBL14264134 0.75 ALDH1A1 (0.71) NPY5RMEN1KMT2A
SCHEMBL14264133 0.75 ALDH1A1 (0.66) NPY5RMEN1KMT2A
SCHEMBL29664801 0.73 ALDH1A1 (0.49) ADORA2ACTSKMEN1KMT2A
SCHEMBL6235242 0.73 CTSK (0.76) ADORA2ACTSKMEN1KMT2A
SCHEMBL9480610 0.72 RAB9A (0.61) KDRMERTKNPY5RMEN1KMT2A
SCHEMBL10099686 0.72 KCNH3 (0.77) ADORA2AADORA2BMERTKNPY5RMEN1
SCHEMBL10073747 0.72 KCNH3 (0.77) ADORA2AADORA2BMERTKNPY5RMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011703-A1 2-CYANO-1,3,5-TRIAZINE-4,6-DIAMINE DERIVATIVES AKZO NOBEL N.V. (NL) 2005-02-10 WO disclosed