SCHEMBL6237989

SCHEMBL6237989

COc1cccc(COCCNCC(N)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.49
AGXT P21549 2/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HTR1A P08908 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
SPHK2 Q9NRA0 1/20 0.46
SPHK1 Q9NYA1 1/20 0.46
MTNR1A P48039 3/20 0.46
MTNR1B P49286 2/20 0.46
TSHR P16473 1/20 0.45
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5099389 0.82 MTNR1A (0.65) MEN1KMT2AALDH1A1KDM4EMTNR1A
SCHEMBL6240427 0.82 CYP3A4 (0.46) IDO1AGXTALDH1A1KDM4EHTR1A
SCHEMBL6237993 0.81 CHRM2 (0.55) IDO1AGXTMEN1KMT2AALDH1A1
SCHEMBL4584070 0.81 MEN1 (0.65) MEN1KMT2AALDH1A1KDM4EHTT
SCHEMBL6239312 0.81 SMN1; SMN2 (0.52) MEN1KMT2AHTTSMN1; SMN2HTR1A
SCHEMBL6239811 0.80 SIRT2 (0.49) MEN1KMT2AALDH1A1TSHR
SCHEMBL17072667 0.76 KDM4E (0.59) ALDH1A1KDM4ESMN1; SMN2SPHK2SPHK1
SCHEMBL6237705 0.75 RAB9A (0.45) AGXTALDH1A1HTTSMN1; SMN2SPHK2
SCHEMBL6235212 0.75 IDO1 (0.45) IDO1MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL2970007 0.74 IDO1 (0.59) IDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011697-A2 SULFONAMIDE DERIVATIVES WITH ACTIVITY ON PROTEIN KINASE A AND B ASTEX THERAPEUTICS LIMITED (GB) 2005-02-10 WO disclosed