SCHEMBL625188

SCHEMBL625188

CC(C)(C)OC(=O)NCC1CCN(c2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
MAPT P10636 13/20 0.42
THRB P10828 3/20 0.41
GAA P10253 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41
PIK3CA P42336 1/20 0.40
LMNA P02545 1/20 0.39
MAP3K12 Q12852 1/20 0.39
ACACB O00763 1/20 0.39
ACACA Q13085 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625132 0.88 CKS1B (0.42) CKS1BSKP1SKP2MAPTTHRB
SCHEMBL625187 0.88 PIK3CA (0.47) CKS1BSKP1SKP2SIRT2SIRT1
SCHEMBL624991 0.85 SYK (0.45) CKS1BSKP1SKP2PIK3CAMAP3K12
SCHEMBL626169 0.84 MAP3K12 (0.41) MAPTTHRBGAAPIK3CALMNA
SCHEMBL624412 0.83 MAP3K12 (0.45) MAPTPIK3CAMAP3K12
SCHEMBL626106 0.82 THRB (0.49) MAPTTHRBGAAPIK3CA
SCHEMBL625422 0.82 PIK3CA (0.42) CKS1BSKP1SKP2MAPTTHRB
SCHEMBL625621 0.81 MAP3K12 (0.46) MAPTPIK3CAMAP3K12
SCHEMBL627373 0.80 MAP3K12 (0.46) MAPTTHRBPIK3CAMAP3K12
SCHEMBL626464 0.80 MAPT (0.47) MAPTTHRBGAAPIK3CALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed