SCHEMBL625331

SCHEMBL625331

CN(CC1CCN(C(=O)OC(C)(C)C)CC1)c1nn2cc(-c3cccc(OC(F)(F)F)c3)nc2s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 5/20 0.45
GPR119 Q8TDV5 3/20 0.40
GLS O94925 1/20 0.40
ABHD6 Q9BV23 1/20 0.38
DAGLA Q9Y4D2 1/20 0.38
KCNH2 Q12809 2/20 0.37
PIM2 Q9P1W9 1/20 0.37
HPGD P15428 3/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
F2RL3 Q96RI0 1/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624434 0.88 JAK2 (0.48) GPR119HPGDMAPTKDM4EALDH1A1
SCHEMBL624009 0.84 PIM1 (0.44) PIM1KCNH2PIM2MAPTF2RL3
SCHEMBL625330 0.84 PIM1 (0.52) PIM1KCNH2PIM2
SCHEMBL624533 0.84 PIM1 (0.53) PIM1GLSKCNH2PIM2MAPT
SCHEMBL623580 0.82 PIM1 (0.40) PIM1GLSKCNH2PIM2MAPT
SCHEMBL623873 0.82 IDH1 (0.44) PIM1GPR119ABHD6DAGLAKCNH2
SCHEMBL627188 0.78 GPR119 (0.40) GPR119GLSHPGDMAPTKDM4E
SCHEMBL625512 0.77 THRB (0.44) PIM1MAPTF2RL3GAA
SCHEMBL624454 0.77 PIM1 (0.45) PIM1GPR119ABHD6DAGLAKCNH2
SCHEMBL623029 0.77 ACKR3 (0.51) PIM1ABHD6DAGLAF2RL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed