SCHEMBL625673

SCHEMBL625673

CN1CCC(CNc2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 16/20 0.48
PIK3CA P42336 2/20 0.41
MAP4K1 Q92918 1/20 0.40
F2RL3 Q96RI0 1/20 0.39
DLK1 P80370 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626702 0.89 MAP3K12 (0.43) MAP3K12PIK3CAF2RL3DLK1
SCHEMBL627611 0.89 MAP3K12 (0.43) MAP3K12PIK3CAF2RL3DLK1
SCHEMBL626582 0.87 PIK3CA (0.42) MAP3K12PIK3CA
SCHEMBL624985 0.86 KDM4E (0.40) MAP3K12PIK3CAMAP4K1
SCHEMBL625672 0.84 PIK3CA (0.53) MAP3K12PIK3CA
SCHEMBL626269 0.80 F2RL3 (0.44) MAP3K12PIK3CAF2RL3
SCHEMBL626289 0.79 PIK3CA (0.42) MAP3K12PIK3CAF2RL3
SCHEMBL12474086 0.79 PIK3CA (0.47) MAP3K12PIK3CAF2RL3
SCHEMBL626145 0.79 F2RL3 (0.43) MAP3K12PIK3CAF2RL3
SCHEMBL626169 0.77 MAP3K12 (0.41) MAP3K12PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed