SCHEMBL625723

SCHEMBL625723

O=C(O)c1sc(Br)nc1Br

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
GPR35 Q9HC97 9/20 0.38
SMN1; SMN2 Q16637 2/20 0.33
DAO P14920 1/20 0.33
PTPN1 P18031 1/20 0.33
KDM4E B2RXH2 4/20 0.32
RAB9A P51151 2/20 0.32
GAA P10253 1/20 0.32
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
PKM P14618 1/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626686 0.78 GAA (0.35) KDM4ERAB9AGAACDC7DBF4
SCHEMBL29877075 0.76 ALDH1A1 (0.45) ALDH1A1HPGDTSHRGPR35SMN1; SMN2
SCHEMBL241856 0.76 ALDH1A1 (0.61) ALDH1A1HPGDTSHRGPR35SMN1; SMN2
SCHEMBL20894398 0.74 ALDH1A1 (0.36) ALDH1A1HPGDTSHRGPR35SMN1; SMN2
SCHEMBL18059154 0.74 ALDH1A1 (0.32) ALDH1A1HPGDTSHRGPR35PTPN1
SCHEMBL16346305 0.74 GPR35 (0.42) ALDH1A1HPGDTSHRGPR35SMN1; SMN2
SCHEMBL14036968 0.73 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2KDM4ERAB9ANPC1
SCHEMBL18173828 0.73 GPR35 (0.42) ALDH1A1HPGDTSHRGPR35POLB
SCHEMBL13534398 0.73 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2KDM4ERAB9A
SCHEMBL622999 0.73 HSD17B10 (0.47) ALDH1A1HPGDTSHRKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 81 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12540134-B2 Inhibitors of adrenoreceptor ADRAC2 BAYER AKTIENGESELLSCHAFT (DE) 2026-02-03 US disclosed
CN-120136863-A Adrenergic receptor ADRAC2 antagonists 拜耳公司 2025-06-13 CN disclosed
CN-120025327-A Adrenergic receptor ADRAC2 antagonists 拜耳公司 2025-05-23 CN disclosed
CN-120025328-A Adrenergic receptor ADRAC2 antagonists 拜耳公司 2025-05-23 CN disclosed
EP-4532485-A1 TYK2 INHIBITORS AND USES THEREOF Sudo Biosciences Limited (GB) 2025-04-09 EP disclosed
WO-2025068514-A1 SUBSTITUTED HETEROCYCLIC CARBOXAMINDES AND USE THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2025-04-03 WO disclosed
CN-114929694-B Adrenergic receptor ADRAC2 antagonists 拜耳公司 2025-02-07 CN disclosed
WO-2024199524-A1 COMPOUND AS PKMYT1 INHIBITOR 江苏星盛新辉医药有限公司 2024-10-03 WO disclosed
US-20240189309-A1 TYK2 INHIBITORS AND USES THEREOF SUDO BIOSCIENCES LIMITED (GB) 2024-06-13 US disclosed
US-20240000767-A1 COMBINATION OF AN ALPHA2-ADRENOCEPTOR SUBTYPE C (ALPHA-2C) ANTAGONIST WITH A TASK1/3 CHANNEL BLOCKER FOR THE TREATMENT OF SLEEP APNEA BAYER AKTIENGESELLSCHAFT (DE) 2024-01-04 US disclosed
US-7323482-B2 Thiazolyl-based compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-01-29 US disclosed
WO-2007096315-A1 4-PHENYL-THIAZOLE-5-CARBOXYLIC ACIDS AND 4-PHENYL-THIAZOLE-5-CARBOXYLIC ACID AMIDES AS PLK1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-30 WO disclosed
WO-2007096315-A1 4-PHENYL-THIAZOLE-5-CARBOXYLIC ACIDS AND 4-PHENYL-THIAZOLE-5-CARBOXYLIC ACID AMIDES AS PLK1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-30 WO disclosed
US-20070203210-A1 Thiazolyl-benzimidazoles BOYLAN JOHN FREDERICK 2007-08-30 US disclosed
US-20070203210-A1 Thiazolyl-benzimidazoles BOYLAN JOHN FREDERICK 2007-08-30 US disclosed
US-20070203210-A1 Thiazolyl-benzimidazoles BOYLAN JOHN FREDERICK 2007-08-30 US disclosed
US-20070093537-A1 Thiazolyl-based compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-04-26 US disclosed
US-20070093537-A1 Thiazolyl-based compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-04-26 US disclosed
US-7169771-B2 Thiazolyl-based compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-30 US disclosed
US-7169771-B2 Thiazolyl-based compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240189309-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK2, JAK1 ALDH1A1 4745/4885HPGD 4028/4885TSHR 2031/4885
US-20070203210-A1 Thiazolyl-benzimidazoles CYP3A7, CYP2C19, CYP3A5 ALDH1A1 100/4885HPGD 1891/4885TSHR 876/4885
US-20240000767-A1 COMBINATION OF AN ALPHA2-ADRENOCEPTOR SUBTYPE C (ALPHA-2C) ANTAGONIST WITH A TASK1/3 CHANNEL BLOCKER FOR THE TREATMENT OF SLEEP APNEA ADRA2C, ADRB2, CHRNA2 ALDH1A1 680/4885HPGD 3134/4885TSHR 2427/4885
US-12540134-B2 Inhibitors of adrenoreceptor ADRAC2 ADRA2C, ADRB3, ADRB2 ALDH1A1 2100/4885HPGD 3170/4885TSHR 613/4885
US-20070093537-A1 Thiazolyl-based compounds useful as kinase inhibitors MAP3K1, MAPK1, MAP3K5 ALDH1A1 1540/4885HPGD 1677/4885TSHR 1104/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.