SCHEMBL627015

SCHEMBL627015

CC(C)(C)OC(=O)N1CCN(CCNc2nn3cc(I)nc3s2)CC1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 10/20 0.61
KMT5A Q9NQR1 1/20 0.42
TLR8 Q9NR97 1/20 0.41
TGFBR1 P36897 1/20 0.36
TGFBR2 P37173 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
STAT3 P40763 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627067 0.82 KDM4E (0.46) ACKR3
SCHEMBL627884 0.81 CCNA2 (0.50) ACKR3
SCHEMBL627014 0.80 ACKR3 (0.63) ACKR3KMT5ATLR8TGFBR1TGFBR2
SCHEMBL627341 0.79 NAMPT (0.47) ACKR3
SCHEMBL626663 0.78 BCHE (0.42) ACKR3
SCHEMBL623029 0.78 ACKR3 (0.51) ACKR3
SCHEMBL625492 0.77 NAMPT (0.39) ACKR3
SCHEMBL627265 0.77 CKS1B (0.41) ACHE
SCHEMBL31287033 0.73 ACKR3 (0.56) ACKR3KMT5A
SCHEMBL628407 0.71 CYP11B2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed