SCHEMBL6274459

SCHEMBL6274459

NC(=O)c1nccc2c(CO)cccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
ALOX12 P18054 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.41
HTT P42858 2/20 0.37
CYP1A2 P05177 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
PARP10 Q53GL7 1/20 0.36
BRAF P15056 3/20 0.36
LCK P06239 1/20 0.36
MAP2K3 P46734 1/20 0.36
MAP2K6 P52564 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433788 0.79 KDM4E (0.54) KDM4ELMNAMAPTTP53TSHR
SCHEMBL1503132 0.79 KDM4E (0.49) KDM4ELMNAMAPTTSHRL3MBTL1
SCHEMBL9849262 0.74 L3MBTL1 (0.39) KDM4EL3MBTL1NPC1RAB9ABRAF
SCHEMBL27626910 0.74 TTR (0.51) KDM4EL3MBTL1CYP1A2KMT2AMEN1
SCHEMBL9849287 0.72 PLAU (0.40) KDM4EL3MBTL1KMT2AMEN1BRAF
SCHEMBL6989543 0.72 LMNA (0.50) KDM4ELMNAMAPTTP53TSHR
SCHEMBL111310 0.72 CNR2 (0.53) KDM4ELMNAMAPTTP53TSHR
SCHEMBL29358323 0.72 CNR2 (0.53) KDM4ELMNAMAPTTP53TSHR
SCHEMBL9849291 0.71 PLAU (0.39) KDM4EL3MBTL1KMT2AMEN1BRAF
SCHEMBL3034972 0.71 APOBEC3G (0.48) KDM4ELMNAMAPTTP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005121094-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTI-HIV-AGENTS PFIZER LIMITED (GB) 2005-12-22 WO disclosed