SCHEMBL6284373

SCHEMBL6284373

COc1ccc(C2C(=O)Nc3ccccc3CN2Cc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
ALDH1A1 P00352 4/20 0.47
HSD17B10 Q99714 1/20 0.47
RORC P51449 1/20 0.46
SIGMAR1 Q99720 3/20 0.44
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
TSHR P16473 2/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6287411 0.85 MEN1 (0.42) KMT2AMEN1ALDH1A1RORCCYP3A4
SCHEMBL6284400 0.75 KDM4E (0.45) ALDH1A1HSD17B10RORCTSHRKDM4E
SCHEMBL6280465 0.75 ALDH1A1 (0.43) KMT2AMEN1ALDH1A1HSD17B10POLB
SCHEMBL18719826 0.71 SIGMAR1 (0.59) KMT2AMEN1CRHBPCRHR2RORC
SCHEMBL6280031 0.71 DDB1 (0.54) KMT2AMEN1ALDH1A1HSD17B10RAB9A
Iodide SCHEMBL27305201 0.70 HDAC8 (0.60) RORCSIGMAR1
SCHEMBL6289026 0.69 ACHE (0.42) ALDH1A1POLBKDM4EMAPT
SCHEMBL6289025 0.69 ACHE (0.42) ALDH1A1POLBKDM4EMAPT
SCHEMBL6286303 0.69 CALCRL (0.38) KMT2AMEN1ALDH1A1HSD17B10KDM4E
SCHEMBL6166562 0.68 CHRM3 (0.55) KMT2AMEN1ALDH1A1SIGMAR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6927294-B1 Nitrogen-containing heterocycles UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2005-08-09 US disclosed