SCHEMBL6315112

SCHEMBL6315112

CSc1nc(N)nc(CN(Cc2ccccc2)C(C)C)n1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.52
HSP90AB1 P08238 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.37
PPARG P37231 1/20 0.35
RAB9A P51151 1/20 0.34
DHFR P00374 2/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307180 0.83 HSP90AA1 (0.57) HSP90AA1HSP90AB1SMN1; SMN2PPARGRAB9A
SCHEMBL6315157 0.77 HSP90AA1 (0.60) HSP90AA1HSP90AB1PPARGDHFRADORA2A
SCHEMBL6309423 0.74 HSP90AA1 (0.57) HSP90AA1HSP90AB1DHFRADORA2AADORA1
SCHEMBL3635237 0.73 TSHR (0.54) SMN1; SMN2SIGMAR1TSHR
SCHEMBL26317585 0.73 NPC1 (0.56) SMN1; SMN2RAB9AADORA2A
SCHEMBL21530452 0.72 ALDH1A1 (0.48) SMN1; SMN2RAB9AADORA2A
SCHEMBL3160936 0.71 MAOB (0.52) RAB9AADORA2AADORA1SIGMAR1TSHR
SCHEMBL6315317 0.70 HSP90AA1 (0.59) HSP90AA1HSP90AB1SMN1; SMN2RAB9AADORA2A
SCHEMBL6315250 0.69 NPC1 (0.71) HSP90AA1HSP90AB1SMN1; SMN2RAB9A
SCHEMBL31612527 0.66 CYP2C19 (0.55) SMN1; SMN2SIGMAR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6919339-B2 ABCA-1 elevating compounds CV THEAPEUTICS, INC. (US) 2005-07-19 US disclosed
EP-1341773-A2 SUBSTITUTED 1,3,5-TRIAZINES AND PYRIMIDINES AS ABCA-1 ELEVATING COMPOUNDS AGAINST CORONARY ARTERY DISEASE OR ATHEROSCLEROSIS CV THERAPEUTICS, INC. (US) 2003-09-10 EP disclosed
US-20020128266-A1 ABCA-1 elevating compounds CV THERAPEUTICS, INC. 2002-09-12 US disclosed
WO-2002046172-A2 SUBSTITUTED 1, 3, 5-TRIAZINES AND PYRIMIDINES AS ABCA-1 ELEVATING COMPOUNDS AGAINST CORONARY ARTERY DISEASE OR ATHEROSCLEROSIS CV THERAPEUTICS, INC. (US) 2002-06-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020128266-A1 ABCA-1 elevating compounds ABCD3, ABCE1, ABCB4 HSP90AA1 1676/4885HSP90AB1 1191/4885SMN1; SMN2 4558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.