SCHEMBL6338288

SCHEMBL6338288

Nc1ccc(CNCCO)c(N)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
CXCR4 P61073 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
USP28 Q96RU2 1/20 0.35
USP25 Q9UHP3 1/20 0.35
EPHX2 P34913 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
CYP2C9 P11712 1/20 0.35
LMNA P02545 1/20 0.35
PDCD1LG2 Q9BQ51 3/20 0.35
CD274 Q9NZQ7 3/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GSR P00390 1/20 0.34
TSHR P16473 1/20 0.34
STAT3 P40763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6339523 0.98 ALDH1A1 (0.41) MAPK1CXCR4ALDH1A1KMT2ACYP1A2
SCHEMBL6266405 0.85 MAPK1 (0.41) MAPK1ALDH1A1KMT2ACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6855744 0.84 MAPK1 (0.43) MAPK1ALDH1A1KMT2ACYP1A2CYP2D6
SCHEMBL6339754 0.83 CXCR4 (0.42) CXCR4KMT2AEPHX2NR1H4HTT
SCHEMBL16429762 0.82 USP28 (0.49) MAPK1CXCR4ALDH1A1KMT2AUSP28
Hydrochloric Acid SCHEMBL6336207 0.81 CXCR4 (0.41) CXCR4ALDH1A1KMT2AEPHX2NR1H4
SCHEMBL34071 0.80 PRKCI (0.47) MAPK1CYP2D6TSHR
Hydrochloric Acid SCHEMBL28744688 0.79 ACHE (0.49) MAPK1ALDH1A1KMT2ACYP1A2CYP2D6
SCHEMBL13242873 0.79 USP28 (0.41) MAPK1ALDH1A1KMT2ACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL28833709 0.79 ACHE (0.49) MAPK1ALDH1A1KMT2ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936077-B2 1,3-diamino-4-(aminomethyl)—benzene derivatives and colorants containing the said compounds WELLA AG (DE) 2005-08-30 US claimed
EP-1370514-A1 1,3-DIAMINO-4-(AMINOMETHYL)-BENZENE DERIVATIVES AND COLORANTS CONTAINING SAID COMPOUNDS Wella Aktiengesellschaft (DE) 2003-12-17 EP claimed
US-20030172471-A1 1,3-diamino-4-(aminomethyl) - benzene derivatives and colorants containing the said compounds HFC PRESTIGE INTERNATIONAL OPERATIONS SWITZERLAND SÀRL (CH) 2003-09-18 US claimed
WO-2002076923-A1 1,3-DIAMINO-4-(AMINOMETHYL)-BENZENE DERIVATIVES AND COLORANTS CONTAINING SAID COMPOUNDS WELLA AKTIENGESELLSCHAFT (DE) 2002-10-03 WO claimed
US-6936077-B2 1,3-diamino-4-(aminomethyl)—benzene derivatives and colorants containing the said compounds WELLA AG (DE) 2005-08-30 US disclosed
EP-1370514-A1 1,3-DIAMINO-4-(AMINOMETHYL)-BENZENE DERIVATIVES AND COLORANTS CONTAINING SAID COMPOUNDS Wella Aktiengesellschaft (DE) 2003-12-17 EP disclosed
US-20030172471-A1 1,3-diamino-4-(aminomethyl) - benzene derivatives and colorants containing the said compounds HFC PRESTIGE INTERNATIONAL OPERATIONS SWITZERLAND SÀRL (CH) 2003-09-18 US disclosed
WO-2002076923-A1 1,3-DIAMINO-4-(AMINOMETHYL)-BENZENE DERIVATIVES AND COLORANTS CONTAINING SAID COMPOUNDS WELLA AKTIENGESELLSCHAFT (DE) 2002-10-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030172471-A1 1,3-diamino-4-(aminomethyl) - benzene derivatives and colorants containing the said compounds AOC1, DPYD, NDUFB4 MAPK1 150/4885CXCR4 4123/4885ALDH1A1 26/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.