SCHEMBL634753

SCHEMBL634753

Cc1cc(N2C(=O)N(CCCCCN3C(=O)N(c4ccc(NC(=O)O)c(C)c4)C(C)(C)C3=O)C(=O)C2(C)C)ccc1NC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
GFER P55789 1/20 0.37
KMT2A Q03164 4/20 0.37
LMNA P02545 2/20 0.36
MEN1 O00255 2/20 0.34
APOBEC3A P31941 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
FAAH O00519 1/20 0.34
MGLL Q99685 1/20 0.34
TP53 P04637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
USP2 O75604 2/20 0.32
PSMD14 O00487 1/20 0.32
MMP2 P08253 1/20 0.32
GRM1 Q13255 1/20 0.32
GRM4 Q14833 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL634406 0.89 PPARG (0.38) PPARGPPARDPPARAGFERKMT2A
SCHEMBL634752 0.79 AR (0.46) PPARGPPARDPPARA
SCHEMBL633869 0.76 AR (0.47)
SCHEMBL634102 0.68 AR (0.50)
SCHEMBL2091371 0.60 MEN1 (0.71) KMT2ALMNAMEN1TP53ALDH1A1
SCHEMBL8048607 0.60 SLC1A3 (0.53) KMT2AMEN1TP53ALDH1A1GAA
SCHEMBL11118946 0.60 GPR174 (0.59) KMT2AMEN1TP53ALDH1A1GAA
SCHEMBL7571649 0.59 MGLL (0.72) LMNAFAAHMGLLALDH1A1GAA
SCHEMBL4830911 0.59 MAPT (0.49) KMT2ALMNAMEN1TP53ALDH1A1
Fluoride SCHEMBL11786773 0.59 MEN1 (0.69) KMT2ALMNAMEN1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2419422-B1 IMIDAZOLIDINE-2,4-DIONE DERIVATIVES AND USE THEREOF AS A MEDICAMENT IPSEN PHARMA SAS (FR) 2014-10-15 EP disclosed
US-8624037-B2 Imidazolidine-2,4-dione derivatives and use thereof as a medicament IPSEN PHARMA S.A.S. (FR) 2014-01-07 US disclosed
EP-2419422-A1 IMIDAZOLIDINE-2,4-DIONE DERIVATIVES AND USE THEREOF AS A MEDICAMENT IPSEN PHARMA S.A.S. (FR) 2012-02-22 EP disclosed
WO-2010119194-A1 IMIDAZOLIDINE-2,4-DIONE DERIVATIVES AND USE THEREOF AS A MEDICAMENT IPSEN PHARMA S.A.S. (FR) 2010-10-21 WO disclosed