SCHEMBL6403148

SCHEMBL6403148

C[n+]1cccc2c(N)cccc21

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
CYP3A4 P08684 2/20 0.48
HPGD P15428 2/20 0.48
TSHR P16473 2/20 0.48
HSD17B10 Q99714 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
NQO2 P16083 2/20 0.42
ACHE P22303 1/20 0.42
KEAP1 Q14145 1/20 0.41
RAB9A P51151 1/20 0.41
RCE1 Q9Y256 1/20 0.41
CHAT P28329 1/20 0.40
NR4A2 P43354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL29561357 0.98 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDTSHRHSD17B10
Iodide SCHEMBL21814312 0.98 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL13829247 0.85 RAB9A (0.50) ACHERAB9ARCE1CHAT
SCHEMBL12529937 0.77 NQO2 (0.60) ALDH1A1NQO2ACHERAB9ARCE1
SCHEMBL8754514 0.77 NQO2 (0.43) ALDH1A1NQO2ACHERAB9ARCE1
SCHEMBL19121786 0.77 CYP2A6 (0.50) ALDH1A1NQO2RAB9ARCE1CHAT
SCHEMBL9331979 0.75 ALDH1A1 (0.48) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL1261956 0.75 ALDH1A1 (0.48) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL9332720 0.75 MAPT (0.51) HPGDTSHRHSD17B10TDP1NQO2
SCHEMBL24373985 0.72 NQO2 (0.40) CYP3A4HPGDTSHRNQO2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12071409-B2 Quinoline derived small molecule inhibitors of nicotinamide N-methyltransferase (NNMT) and uses thereof THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS (US) 2024-08-27 US disclosed
US-20230107256-A1 QUINOLINE DERIVED SMALL MOLECULE INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE (NNMT) AND USES THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2023-04-06 US disclosed
US-11401243-B2 Quinoline derived small molecule inhibitors of nicotinamide N-methyltransferase (NNMT) and uses thereof THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-08-02 US disclosed
US-20200102274-A1 QUINOLINE DERIVED SMALL MOLECULE INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE (NNMT) AND USES THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2020-04-02 US disclosed
US-20050171195-A1 P2X7 antagonists for treating neuropathic pain ABBOTT LABORATORIES 2005-08-04 US disclosed
EP-0315997-B1 Cephalosporin compounds and antibacterial agents MEIJI SEIKA KAISHA (JP) 1994-04-20 EP disclosed
US-5028601-A Substituted with an amino thiazole group and a dihydroxy-pyridone group MEIJI SAIKA KAISHA, LTD. (JP) 1991-07-02 US disclosed
US-4971961-A ANTIBIOTICS AS BACTERICIDES AGAINST PSEUDOMONAS MEIJI SEIKA KAISHA, LTD. (JP) 1990-11-20 US disclosed
EP-0289002-A2 Novel cephalosporin compounds and antibacterial agents MEIJI SEIKA KAISHA LTD. (JP) 1988-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171195-A1 P2X7 antagonists for treating neuropathic pain P2RX3, P2RX7, P2RX1 ALDH1A1 1730/4885CYP3A4 3130/4885HPGD 1153/4885
US-20200102274-A1 QUINOLINE DERIVED SMALL MOLECULE INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE (NNMT) AND USES THEREOF NNMT, NAMPT, NNT ALDH1A1 459/4885CYP3A4 823/4885HPGD 124/4885
US-20230107256-A1 QUINOLINE DERIVED SMALL MOLECULE INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE (NNMT) AND USES THEREOF NNMT, NAMPT, NNT ALDH1A1 755/4885CYP3A4 875/4885HPGD 140/4885
US-12071409-B2 Quinoline derived small molecule inhibitors of nicotinamide N-methyltransferase (NNMT) and uses thereof NNMT, NAMPT, NNT ALDH1A1 755/4885CYP3A4 875/4885HPGD 140/4885
US-11401243-B2 Quinoline derived small molecule inhibitors of nicotinamide N-methyltransferase (NNMT) and uses thereof NNMT, NAMPT, NNT ALDH1A1 459/4885CYP3A4 823/4885HPGD 124/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.