SCHEMBL6409750

SCHEMBL6409750

O=C(O)OC1=NOC2(CCN(C(=O)c3ccc(Br)cc3)CC2)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.47
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
NEK2 P51955 1/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 1/20 0.40
MGLL Q99685 1/20 0.40
HSD11B1 P28845 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6410146 0.86 TSHR (0.43) HPGDNEK2TSHRPOLBHDAC3
SCHEMBL6418195 0.86 POLB (0.55) HPGDTSHRPOLBKMT2ASMN1; SMN2
SCHEMBL6410215 0.85 SLC6A7 (0.42) HPGDTSHRPOLBMGLLKMT2A
SCHEMBL6410053 0.85 MGLL (0.42) HPGDTSHRPOLBMGLLHDAC3
SCHEMBL6409864 0.84 KMT2A (0.43) HPGDNEK2POLBHDAC3HDAC4
SCHEMBL6410851 0.83 HSD11B1 (0.47) MGLLHSD11B1
SCHEMBL2402430 0.83 HPGD (0.49) HPGDCA12CA1CA2CA7
SCHEMBL6411763 0.82 EPHX2 (0.38) HPGDTSHRPOLBMGLLHDAC3
SCHEMBL6413167 0.80 FPR3 (0.37) HPGDCA12CA1CA2CA7
SCHEMBL6415785 0.80 HTR1A (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP disclosed