SCHEMBL6419294

SCHEMBL6419294

CCC(COC(=O)C(=O)On1cnc2c1CCN(C(=O)O)C2)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.37
GAA P10253 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 1/20 0.34
P2RX7 Q99572 4/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
PKM P14618 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423522 0.83 PDK2 (0.39) PDK2P2RX7PTGDR2
SCHEMBL6420064 0.80 GRIN2B (0.38) PDK2GAAALDH1A1KDM4EP2RX7
SCHEMBL6419465 0.79 PDK2 (0.36) PDK2P2RX7PTGDR2CHRM2CHRM4
SCHEMBL6422824 0.78 CHRM5 (0.41) PDK2GAAALDH1A1P2RX7PTGDR2
SCHEMBL6422607 0.78 P2RX7 (0.43) PDK2ALDH1A1P2RX7PTGDR2
SCHEMBL6422956 0.77 CHRM5 (0.42) ALDH1A1KDM4ECHRM5CHRM1
SCHEMBL6420512 0.76 GRIN2B (0.40) ALDH1A1CHRM5CHRM1
SCHEMBL6423885 0.76 PTGDR2 (0.37) PDK2P2RX7PTGDR2
SCHEMBL6423530 0.76 PTGDR2 (0.36) PDK2ALDH1A1P2RX7PTGDR2
SCHEMBL6420047 0.76 PTGDR2 (0.37) PDK2P2RX7PTGDR2CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6908926-B1 Substituted imidazoles, their preparation and use NOVO NORDISK A/S (DK) 2005-06-21 US disclosed
EP-1173438-A1 SUBSTITUTED IMIDAZOLES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2002-01-23 EP disclosed
WO-2000063208-A1 SUBSTITUTED IMIDAZOLES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2000-10-26 WO disclosed