SCHEMBL6426403

SCHEMBL6426403

O[C@]1(c2ccc3cc[nH]c3c2)CCN2CCC[C@H]2C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.48
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HSD17B10 Q99714 3/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
CHRNA7 P36544 2/20 0.37
HTR3A P46098 1/20 0.37
ALOX12 P18054 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
AHR P35869 1/20 0.35
TYR P14679 1/20 0.35
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRL1 P41146 2/20 0.34
CCR1 P32246 4/20 0.34
SLC18A3 Q16572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6740915 1.00 HTR6 (0.48) HTR6KDM4EALDH1A1HSD17B10MAPT
SCHEMBL7997497 0.74 HTR6 (0.46) HTR6KDM4EALDH1A1MAPTCCR1
SCHEMBL6744625 0.73 AHR (0.42) KDM4EALDH1A1HSD17B10HPGDCHRNA7
SCHEMBL7006323 0.73 CYP1A2 (0.55) MAPT
SCHEMBL7005001 0.71 HTR1A (0.47) HTR6HTR3A
SCHEMBL7501279 0.71 HTR6 (0.44) HTR6ALDH1A1CHRNA7HTR3ACNR2
SCHEMBL7006270 0.70 HTR1B (0.58) HTR6
SCHEMBL7006286 0.70 HTR1B (0.58) HTR6
SCHEMBL7006099 0.69 SLC6A4 (0.53)
SCHEMBL7010984 0.69 SLC6A4 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897215-B1 Compounds having 5-HT6 receptor antagonist activity NPS ALLELIX CORP. (CA) 2005-05-24 US disclosed
WO-2001032660-A1 COMPOUNDS HAVING 5-HT6 RECEPTOR ANTAGONIST ACTIVITY NPS ALLELIX CORP. (US) 2001-05-10 WO disclosed