SCHEMBL6443471

SCHEMBL6443471

N#CCCNC(=O)C(CNC(=O)c1ccccc1F)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
CTSS P25774 2/20 0.44
CTSK P43235 2/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ATM Q13315 1/20 0.42
CTSL P07711 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 2/20 0.41
HPGD P15428 1/20 0.41
KDM4E B2RXH2 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
ALDH1A1 P00352 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HDAC7 Q8WUI4 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447527 0.92 LMNA (0.41) RAB9ANPC1CTSSCTSKMEN1
SCHEMBL6443484 0.89 CTSK (0.55) RAB9ANPC1CTSSCTSKMEN1
SCHEMBL6448077 0.88 KDM4E (0.54) RAB9ANPC1CTSSCTSKMEN1
SCHEMBL6447483 0.87 ATM (0.49) RAB9ANPC1CTSSCTSKMEN1
SCHEMBL6443588 0.84 NPC1 (0.51) RAB9ANPC1CTSSCTSKCTSL
SCHEMBL6472461 0.83 CTSD (0.46) RAB9ANPC1CTSSCTSKMEN1
SCHEMBL6442799 0.83 CTSK (0.54) RAB9ANPC1CTSSCTSKMEN1
SCHEMBL30827958 0.82 NPC1 (0.60) RAB9ANPC1MEN1KMT2ALMNA
SCHEMBL6825007 0.82 KDM4E (0.47) CTSSCTSKMEN1KMT2ACTSL
SCHEMBL6822581 0.81 GAA (0.43) RAB9ANPC1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed