SCHEMBL6443588

SCHEMBL6443588

N#CCCNC(=O)C(CNC(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CTSK P43235 7/20 0.48
CTSS P25774 5/20 0.48
EPHX2 P34913 2/20 0.48
CTSL P07711 7/20 0.45
CTSB P07858 2/20 0.45
POLB P06746 1/20 0.43
GAA P10253 1/20 0.41
KDM4A O75164 1/20 0.41
GUSB P08236 1/20 0.40
GPR139 Q6DWJ6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443745 0.93 CTSS (0.47) NPC1RAB9ASMN1; SMN2CTSKCTSS
SCHEMBL6442019 0.90 CTSS (0.42) NPC1RAB9ASMN1; SMN2CTSKCTSS
SCHEMBL5517758 0.88 CTSK (0.61) NPC1RAB9ASMN1; SMN2CTSKCTSS
SCHEMBL6445311 0.88 ALDH1A1 (0.47) SMN1; SMN2CTSKCTSSEPHX2CTSL
SCHEMBL6447322 0.87 CTSK (0.42) NPC1RAB9ASMN1; SMN2CTSKCTSS
SCHEMBL6446599 0.87 GUSB (0.43) NPC1RAB9ASMN1; SMN2CTSKCTSS
SCHEMBL6448077 0.86 KDM4E (0.54) NPC1RAB9ACTSKCTSSCTSL
SCHEMBL6444047 0.86 CTSL (0.53) NPC1SMN1; SMN2CTSLPOLBGPR139
SCHEMBL6443471 0.84 RAB9A (0.46) NPC1RAB9ASMN1; SMN2CTSKCTSS
SCHEMBL6445366 0.83 CTSS (0.47) CTSKCTSSCTSLCTSBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed