SCHEMBL6442019

SCHEMBL6442019

N#CCCNC(=O)C(CNC(=O)c1ccc(CCl)cc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.42
CTSK P43235 6/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4A O75164 1/20 0.41
CTSL P07711 6/20 0.40
GUSB P08236 1/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
EPHX2 P34913 1/20 0.39
CTSB P07858 3/20 0.38
TPSAB1 Q15661 1/20 0.37
CYP24A1 Q07973 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443632 0.90 SFN (0.42) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6444782 0.90 CTSK (0.53) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6443588 0.90 NPC1 (0.51) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6446599 0.88 GUSB (0.43) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6446797 0.88 CTSS (0.43) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6443745 0.83 CTSS (0.47) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6445311 0.83 ALDH1A1 (0.47) CTSSCTSKSMN1; SMN2CTSLPOLB
SCHEMBL6443534 0.81 HDAC6 (0.37) CTSSCTSKSMN1; SMN2CTSLGUSB
SCHEMBL6446405 0.81 CTSL (0.50) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6445190 0.80 GUSB (0.40) CTSSCTSKKDM4ACTSLGUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed