SCHEMBL6443541

SCHEMBL6443541

CCN(C#N)C(=O)C(Cc1ccc2ccccc2c1)NC(=O)c1cccs1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.51
CTSC P53634 1/20 0.50
CTSB P07858 4/20 0.47
CTSS P25774 4/20 0.47
CTSK P43235 2/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
RAB9A P51151 2/20 0.42
PIN1 Q13526 2/20 0.42
HSPA5 P11021 3/20 0.42
CA2 P00918 1/20 0.42
HSPA1A P0DMV8 1/20 0.42
HSPA9 P38646 1/20 0.42
HSPA2 P54652 1/20 0.42
MME P08473 2/20 0.41
ACE P12821 2/20 0.41
CPA1 P15085 1/20 0.41
ACE2 Q9BYF1 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443368 0.88 CTSL (0.53) CTSLCTSCCTSBCTSSCTSK
SCHEMBL6442766 0.88 CTSL (0.65) CTSLCTSCCTSBCTSSCTSK
SCHEMBL6818989 0.86 CTSL (0.54) CTSLCTSBCTSSCTSKRAB9A
SCHEMBL6020522 0.86 CTSL (0.60) CTSLCTSBCTSSCTSKMMP9
SCHEMBL6021205 0.84 MMP9 (0.53) CTSLCTSBCTSSCTSKMMP9
SCHEMBL6020743 0.84 MMP9 (0.53) CTSLCTSCCTSBCTSSCTSK
SCHEMBL6021440 0.83 CTSB (0.53) CTSLCTSBCTSSCTSKMMP9
SCHEMBL6021084 0.83 CTSS (0.50) CTSLCTSCCTSBCTSSCTSK
SCHEMBL6020865 0.82 CTSB (0.47) CTSLCTSBCTSSCTSKMMP9
SCHEMBL6019790 0.82 CTSB (0.56) CTSLCTSBCTSSCTSKMMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed