SCHEMBL6446599

SCHEMBL6446599

N#CCCNC(=O)C(CNC(=O)c1cccc(CCl)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GUSB P08236 1/20 0.43
CTSK P43235 7/20 0.43
CTSS P25774 6/20 0.43
CTSL P07711 6/20 0.43
KDM4A O75164 1/20 0.41
POLB P06746 1/20 0.40
F10 P00742 1/20 0.40
PRSS1 P07477 1/20 0.40
CTSB P07858 3/20 0.39
CTSV O60911 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445190 0.92 GUSB (0.40) GUSBCTSKCTSSCTSLKDM4A
SCHEMBL6447506 0.90 CTSL (0.53) CTSKCTSSCTSLCTSBCTSV
SCHEMBL6446578 0.89 ATM (0.41) GUSBCTSKCTSSCTSLCTSB
SCHEMBL6442019 0.88 CTSS (0.42) GUSBCTSKCTSSCTSLKDM4A
SCHEMBL6443588 0.87 NPC1 (0.51) GUSBCTSKCTSSCTSLKDM4A
SCHEMBL6822562 0.83 CTSK (0.47) CTSKCTSSCTSLCTSBCTSV
SCHEMBL6444047 0.82 CTSL (0.53) CTSLPOLBNPC1SMN1; SMN2GPR139
SCHEMBL6446480 0.82 GUSB (0.36) GUSBCTSKCTSSCTSLCTSB
SCHEMBL6446816 0.82 GAA (0.40) GUSBCTSKCTSSCTSLCTSB
SCHEMBL6443755 0.81 GAA (0.40) GUSBCTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed