SCHEMBL6444201

SCHEMBL6444201

N#CCCNC(=O)C(CNC(=O)c1cccc(C(F)(F)F)c1)c1ccc2ccccc2c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.47
POLB P06746 2/20 0.45
ALDH1A1 P00352 1/20 0.45
KAT6A Q92794 1/20 0.44
ATM Q13315 1/20 0.43
GPR139 Q6DWJ6 1/20 0.43
TACR1 P25103 1/20 0.42
TP53 P04637 1/20 0.41
TP53BP1 Q12888 1/20 0.41
NPC1 O15118 1/20 0.41
DRD2 P14416 1/20 0.41
ADRA1A P35348 1/20 0.41
DRD3 P35462 1/20 0.41
PIN1 Q13526 1/20 0.40
NAMPT P43490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446794 0.91 CTSL (0.58) CTSLPOLBALDH1A1KAT6AATM
SCHEMBL6444047 0.89 CTSL (0.53) CTSLPOLBALDH1A1GPR139TACR1
SCHEMBL6442129 0.88 CTSL (0.49) CTSLPOLBALDH1A1GPR139TACR1
SCHEMBL6447322 0.87 CTSK (0.42) CTSLATMNPC1
SCHEMBL6446578 0.84 ATM (0.41) CTSLATMPIN1
SCHEMBL6446641 0.80 CTSL (0.64) CTSLPOLBALDH1A1GPR139TACR1
SCHEMBL6446797 0.80 CTSS (0.43) CTSLATMNPC1DRD2DRD3
SCHEMBL6447483 0.80 ATM (0.49) CTSLPOLBALDH1A1KAT6AATM
SCHEMBL6020313 0.79 CTSL (0.63) CTSLPIN1
SCHEMBL6822574 0.79 CTSL (0.44) CTSLPOLBALDH1A1GPR139TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed