SCHEMBL6444118

SCHEMBL6444118

N#CCNC(=O)C(CNC(=O)CCC(=O)O)c1ccc(O)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.50
CTSS P25774 7/20 0.50
CYP1A1 P04798 1/20 0.42
CTSL P07711 8/20 0.42
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
CTSB P07858 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443377 0.90 CTSK (0.55) CTSKCTSSCTSLCTSB
SCHEMBL6822727 0.89 CYP1A1 (0.40) CTSKCTSSCYP1A1CTSLESR1
SCHEMBL6446697 0.82 CTSK (0.48) CTSKCTSSCTSLCTSB
SCHEMBL6447927 0.82 CTSK (0.52) CTSKCTSSCTSLESR1ESR2
SCHEMBL6443540 0.80 CTSK (0.60) CTSKCTSSCTSLCTSB
SCHEMBL6442367 0.80 CTSK (0.50) CTSKCTSSCTSLCTSB
SCHEMBL6443393 0.79 CTSK (0.43) CTSKCTSSCTSL
SCHEMBL6445473 0.79 CTSS (0.49) CTSKCTSSCTSLESR1ESR2
SCHEMBL6446467 0.79 CTSK (0.49) CTSKCTSSCTSLCTSB
SCHEMBL6822170 0.79 CTSS (0.49) CTSKCTSSCTSLESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed