SCHEMBL6443377

SCHEMBL6443377

N#CCNC(=O)C(CNC(=O)CCC(=O)O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.55
CTSS P25774 12/20 0.55
CTSL P07711 11/20 0.52
CTSB P07858 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444118 0.90 CTSK (0.50) CTSKCTSSCTSLCTSB
SCHEMBL6443393 0.88 CTSK (0.43) CTSKCTSSCTSL
SCHEMBL6446697 0.87 CTSK (0.48) CTSKCTSSCTSLCTSB
SCHEMBL5526073 0.84 CTSK (0.62) CTSKCTSSCTSLCTSB
SCHEMBL5517758 0.81 CTSK (0.61) CTSKCTSSCTSLCTSB
SCHEMBL6442556 0.81 CTSS (0.58) CTSKCTSSCTSLCTSB
SCHEMBL7872412 0.80 ASAH1 (0.43) CTSSCTSLCTSB
SCHEMBL6446744 0.79 CTSL (0.45) CTSKCTSSCTSLCTSB
SCHEMBL6822727 0.79 CYP1A1 (0.40) CTSKCTSSCTSL
SCHEMBL6445536 0.78 CTSK (0.55) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed