SCHEMBL6443393

SCHEMBL6443393

N#CCCNC(=O)C(CNC(=O)CCC(=O)O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.43
CTSS P25774 3/20 0.43
POLB P06746 1/20 0.41
CTSL P07711 4/20 0.41
KDM4A O75164 1/20 0.40
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ASAH1 Q13510 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ACE P12821 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822727 0.90 CYP1A1 (0.40) CTSKCTSSPOLBCTSLCNR1
SCHEMBL6443377 0.88 CTSK (0.55) CTSKCTSSCTSL
SCHEMBL6822560 0.88 CYP1A2 (0.43) CTSKCTSSCTSLMEN1KMT2A
SCHEMBL6443588 0.82 NPC1 (0.51) CTSKCTSSPOLBCTSLKDM4A
SCHEMBL6445366 0.81 CTSS (0.47) CTSKCTSSPOLBCTSLKDM4A
SCHEMBL6447617 0.81 CTSK (0.37) CTSKCTSSPOLBCTSLCYP2C19
SCHEMBL6443547 0.80 CTSK (0.43) CTSKCTSSPOLBCTSLKDM4A
SCHEMBL6448077 0.79 KDM4E (0.54) CTSKCTSSPOLBCTSLKDM4A
SCHEMBL6447305 0.79 CTSS (0.43) CTSKCTSSPOLBCTSLKDM4A
SCHEMBL6445386 0.79 ALDH1A1 (0.44) CTSKCTSSPOLBCTSLKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed