SCHEMBL6445342

SCHEMBL6445342

CCN(C#N)C(=O)C(CS(C)(=O)=O)NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSB P07858 4/20 0.41
CTSS P25774 3/20 0.41
CTSL P07711 2/20 0.41
CTSK P43235 1/20 0.41
CTSF Q9UBX1 1/20 0.41
CLPP Q16740 2/20 0.41
SCN1A P35498 3/20 0.40
SCN2A Q99250 3/20 0.40
SCN3A Q9NY46 3/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CHRNB2 P17787 2/20 0.38
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
CHRNA4 P43681 2/20 0.38
NPY2R P49146 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6020271 0.89 CTSB (0.43) CTSBCTSSCTSLCTSKCTSF
SCHEMBL6449554 0.87 CTSB (0.45) CTSBCTSSCTSLCTSKCTSF
SCHEMBL6020744 0.86 LMNA (0.40) CTSBCTSSCTSLCTSKCTSF
SCHEMBL6019224 0.85 CTSL (0.55) CTSBCTSSCTSLCTSKCTSF
SCHEMBL6443458 0.85 CTSL (0.47) CTSBCTSSCTSLCTSKCLPP
SCHEMBL6446903 0.85 CLPP (0.43) CTSBCLPPSCN1ASCN2ASCN3A
SCHEMBL6020512 0.82 SMN1; SMN2 (0.43) CTSBCTSSCTSLCTSKCTSF
SCHEMBL6444324 0.81 CTSL (0.50) CTSBCTSSCTSLCTSKCLPP
SCHEMBL6443194 0.79 CTSB (0.51) CTSBCTSSCTSLCTSK
SCHEMBL6021519 0.79 CTSL (0.46) CTSBCTSSCTSLCTSKCTSF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed