Desmethylthiamethoxam

Desmethylthiamethoxam

SCHEMBL6445790

O=[N+]([O-])N=C1NCOCN1Cc1cnc(Cl)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
MAPT P10636 2/20 0.36
LMNA P02545 4/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 2/20 0.33
RECQL P46063 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Desmethylthiamethoxam SCHEMBL7173902 1.00 CHRNB2 (0.40) CHRNB2CHRNA4MAPTLMNAALDH1A1
Desmethylthiamethoxam SCHEMBL6445785 1.00 CHRNB2 (0.40) CHRNB2CHRNA4MAPTLMNAALDH1A1
Imidaclothiz SCHEMBL676082 0.84 CHRNB2 (0.55) CHRNB2CHRNA4MAPTLMNAALDH1A1
Imidaclothiz SCHEMBL238122 0.84 CHRNB2 (0.55) CHRNB2CHRNA4MAPTLMNAALDH1A1
SCHEMBL7982213 0.82 CHRNB2 (0.48) CHRNB2CHRNA4MAPTLMNAALDH1A1
SCHEMBL10062415 0.81 LMNA (0.37) MAPTLMNAALDH1A1GAAKMT2A
SCHEMBL6447070 0.81 CHRNB2 (0.51) CHRNB2CHRNA4MAPTALDH1A1
SCHEMBL6723120 0.81 CHRNB2 (0.51) CHRNB2CHRNA4MAPTALDH1A1
SCHEMBL9866741 0.81 CHRNB2 (0.38) CHRNB2CHRNA4MAPTLMNAALDH1A1
SCHEMBL9866750 0.81 CHRNB2 (0.38) CHRNB2CHRNA4MAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884755-B2 Pesticidal composition SYNGENTA CROP PROTECTION, INC. (US) 2005-04-26 US claimed
US-20030166618-A1 Pesticidal composition SENN ROBERT (CH) 2003-09-04 US claimed
EP-0915656-B1 PESTICIDAL COMPOSITION SYNGENTA PARTICIPATIONS AG (CH) 2003-07-23 EP claimed
EP-0900024-B1 PESTICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2003-06-18 EP claimed
EP-0915656-A1 PESTICIDAL COMPOSITION Novartis AG (CH) 1999-05-19 EP claimed
WO-1997040691-A1 PESTICIDAL COMPOSITION NOVARTIS AG (CH) 1997-11-06 WO claimed
US-6884755-B2 Pesticidal composition SYNGENTA CROP PROTECTION, INC. (US) 2005-04-26 US disclosed
US-20040122227-A1 Cyclic guanidine derivatives and their use as pesticides WAGNER KLAUS (DE) 2004-06-24 US disclosed
US-6683028-B1 Cyclic guanidine derivatives and their use as pesticides BAYER AKTIENGESELLSCHAFT (DE) 2004-01-27 US disclosed
US-20030166618-A1 Pesticidal composition SENN ROBERT (CH) 2003-09-04 US disclosed
EP-0915656-B1 PESTICIDAL COMPOSITION SYNGENTA PARTICIPATIONS AG (CH) 2003-07-23 EP disclosed
EP-0900024-B1 PESTICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2003-06-18 EP disclosed
US-6514954-B1 For controlling insects or representatives of the order Acarina SYNGENTA CROP PROTECTION, INC. 2003-02-04 US disclosed
EP-0915656-A1 PESTICIDAL COMPOSITION Novartis AG (CH) 1999-05-19 EP disclosed
WO-1998006710-A1 SUBSTITUTED 4-NITROIMINO-PERHYDRO-1,3,5-OXADIAZINE DERIVATIVES, THEIR USE AS PESTICIDES AND INTERMEDIATES FOR THEIR PREPARATION NOVARTIS AG (CH) 1998-02-19 WO disclosed
WO-1997040691-A1 PESTICIDAL COMPOSITION NOVARTIS AG (CH) 1997-11-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122227-A1 Cyclic guanidine derivatives and their use as pesticides PRMT1, GUCY1A1, GUCY1A2 CHRNB2 527/4885CHRNA4 440/4885MAPT 4114/4885
US-20030166618-A1 Pesticidal composition TUBA3C, DDT, TUBB3 CHRNB2 453/4885CHRNA4 916/4885MAPT 2830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.