SCHEMBL6446308

SCHEMBL6446308

CC(=O)Nc1ccc(C(=O)NCC(C(=O)NCCC#N)c2ccc(O)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
HTT P42858 1/20 0.42
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 2/20 0.42
NR1H4 Q96RI1 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 2/20 0.42
CA12 O43570 1/20 0.42
BRD4 O60885 1/20 0.42
NR1I2 O75469 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MB P02144 1/20 0.42
CYP1A1 P04798 1/20 0.42
CA3 P07451 1/20 0.42
RARG P13631 1/20 0.42
TSHR P16473 1/20 0.42
ALOX5AP P20292 1/20 0.42
CA4 P22748 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445311 0.91 ALDH1A1 (0.47) SMN1; SMN2HTTALDH1A1CYP3A4NR1H4
SCHEMBL6448227 0.90 CTSS (0.47) SMN1; SMN2HTTALDH1A1CYP3A4NR1H4
SCHEMBL6443466 0.85 MEN1 (0.40) SMN1; SMN2HTTALDH1A1CYP3A4NR1H4
SCHEMBL6443745 0.85 CTSS (0.47) SMN1; SMN2EPHX2CTSSCTSKNPC1
SCHEMBL6443632 0.83 SFN (0.42) SMN1; SMN2MEN1KMT2AMAPTCTSS
SCHEMBL6442110 0.81 CTSS (0.52) SMN1; SMN2HTTALDH1A1MEN1KMT2A
SCHEMBL6442164 0.81 SMN1; SMN2 (0.46) SMN1; SMN2HTTALDH1A1CYP3A4NR1H4
SCHEMBL6442163 0.80 TP53 (0.48) SMN1; SMN2HTTALDH1A1CYP3A4NR1H4
SCHEMBL6019331 0.78 CTSL (0.62) CTSSCTSK
SCHEMBL6446763 0.78 ESR1 (0.41) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed