SCHEMBL6443632

SCHEMBL6443632

N#CCCNC(=O)C(CNC(=O)c1ccc(CCl)cc1)c1ccc(O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SFN P31947 1/20 0.42
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C19 P33261 1/20 0.40
GFER P55789 1/20 0.40
ESRRG P62508 3/20 0.40
CTSL P07711 1/20 0.39
ESRRB O95718 2/20 0.39
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
GUSB P08236 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442019 0.90 CTSS (0.42) RAB9ASMN1; SMN2NPC1CTSLCTSS
SCHEMBL6446405 0.89 CTSL (0.50) SFNRAB9ASMN1; SMN2NPC1CYP1A2
SCHEMBL6445190 0.88 GUSB (0.40) SFNGAACTSLCTSSCTSK
SCHEMBL6443745 0.86 CTSS (0.47) RAB9ASMN1; SMN2NPC1GAACTSL
SCHEMBL6446797 0.85 CTSS (0.43) RAB9ASMN1; SMN2NPC1CTSLCTSS
SCHEMBL6446308 0.83 SMN1; SMN2 (0.42) RAB9ASMN1; SMN2NPC1MAPTCTSS
SCHEMBL6444782 0.80 CTSK (0.53) RAB9ASMN1; SMN2NPC1CTSLCTSS
SCHEMBL6020957 0.79 CTSL (0.64) SFNCTSLCTSSCTSK
SCHEMBL6443588 0.79 NPC1 (0.51) RAB9ASMN1; SMN2NPC1GAACTSL
SCHEMBL6446599 0.79 GUSB (0.43) RAB9ASMN1; SMN2NPC1CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed