SCHEMBL6443745

SCHEMBL6443745

N#CCCNC(=O)C(CNC(=O)c1ccccc1)c1ccc(O)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.47
CTSK P43235 4/20 0.47
CTSL P07711 6/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
CTSB P07858 2/20 0.42
EPHX2 P34913 1/20 0.41
GUSB P08236 2/20 0.40
GAA P10253 1/20 0.38
MIF P14174 1/20 0.37
GLI1 P08151 1/20 0.37
GLI2 P10070 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443588 0.93 NPC1 (0.51) CTSSCTSKCTSLNPC1RAB9A
SCHEMBL6443540 0.89 CTSK (0.60) CTSSCTSKCTSLNPC1RAB9A
SCHEMBL6825007 0.87 KDM4E (0.47) CTSSCTSKCTSLCNR1CNR2
SCHEMBL6443632 0.86 SFN (0.42) CTSSCTSKCTSLNPC1RAB9A
SCHEMBL6447322 0.85 CTSK (0.42) CTSSCTSKCTSLNPC1RAB9A
SCHEMBL6445190 0.85 GUSB (0.40) CTSSCTSKCTSLCTSBGUSB
SCHEMBL6446308 0.85 SMN1; SMN2 (0.42) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6442129 0.84 CTSL (0.49) CTSLNPC1
SCHEMBL6447527 0.84 LMNA (0.41) CTSSCTSKNPC1RAB9ASMN1; SMN2
SCHEMBL6442019 0.83 CTSS (0.42) CTSSCTSKCTSLNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed