SCHEMBL6447040

SCHEMBL6447040

CSC(CNC(=O)c1ccccc1[N+](=O)[O-])C(=O)NCC#N

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.49
ALDH1A1 P00352 5/20 0.48
HPGD P15428 3/20 0.46
HTT P42858 2/20 0.46
LMNA P02545 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CTSB P07858 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
GAA P10253 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443305 0.90 CTSD (0.46) CTSDALDH1A1HPGDHTTLMNA
SCHEMBL6446809 0.84 KDM4E (0.51) HTTMEN1KMT2ACTSBKDM4E
SCHEMBL6445609 0.84 CTSK (0.52) CTSDALDH1A1HPGDHTTLMNA
SCHEMBL6441973 0.83 CTSD (0.48) CTSDALDH1A1HPGDHTTLMNA
SCHEMBL6442378 0.82 GAA (0.47) ALDH1A1HPGDMEN1KMT2ACTSB
SCHEMBL6019589 0.82 CTSL (0.47) CTSDALDH1A1MEN1KMT2ACTSB
SCHEMBL6445280 0.80 CTSK (0.51) CTSDALDH1A1HPGDHTTLMNA
SCHEMBL6447899 0.80 CTSL (0.54) CTSB
SCHEMBL6441987 0.78 CTSK (0.46) CTSDALDH1A1HPGDHTTLMNA
SCHEMBL6020934 0.77 CTSL (0.65) CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed